351.3 🏥 內科專科考前版

351.3.1 Mechanistic Deep Dive

351.3.1.1 Pathophysiology

  • Genetic susceptibility (NOD2/CARD15 in CD)
  • Environmental triggers
  • Dysregulated mucosal immune response
  • Microbiome (dysbiosis)
  • Epithelial barrier dysfunction

351.3.1.2 Th17 + IL-23 Axis

  • Central in IBD inflammation
  • Target for ustekinumab, risankizumab, mirikizumab

351.3.1.3 S1P Receptor in IBD

  • Lymphocyte trafficking
  • Ozanimod, etrasimod inhibit egress from lymph nodes

351.3.1.4 JAK-STAT Pathway

  • Multiple cytokine signaling
  • Tofacitinib, upadacitinib pan-JAK

351.3.2 Recent Trials & Updates

351.3.2.1 LUCENT-1, LUCENT-2 (2023) — Mirikizumab UC

  • IL-23p19 selective
  • FDA approval 2023

351.3.2.2 ADVANCE, MOTIVATE (2022) — Risankizumab CD

  • IL-23p19 selective
  • FDA approval 2022

351.3.2.3 U-EXCEL, U-EXCEED (2023) — Upadacitinib CD

  • JAK inhibitor
  • FDA approval 2023

351.3.2.4 TRUE NORTH (2020) — Ozanimod UC

  • S1P modulator
  • FDA approval 2021

351.3.2.5 ELEVATE UC (2023) — Etrasimod

  • S1P modulator
  • FDA approval 2023

351.3.2.6 CALM Trial — Treat to Target

  • Mucosal healing-driven
  • Improved outcomes

351.3.3 High-Yield Specialist Points

351.3.3.1 Drug Sequencing

  • After biologic failure, next-line consideration
  • Mechanistic differences may help
  • Bio-naive vs bio-experienced have different responses

351.3.3.2 Antibody Levels + Drug Monitoring

  • Infliximab levels + anti-drug antibodies
  • Personalized dosing
  • ↑ Doses for low levels + neutralizing antibodies

351.3.3.3 Vaccination Pre-Biologic

  • Live vaccines avoided
  • Inactivated: flu, pneumococcal, HBV
  • Document immunity

351.3.3.4 Pregnancy + Biologics

  • Maintain TNF inhibitors through 3rd trimester (last dose 4-6 weeks pre-delivery for newer)
  • Vedolizumab: less placental transfer
  • Avoid live vaccines in infant first 6-12 months

351.3.3.5 Anti-TNF Side Effects

  • Infections (TB reactivation — screen)
  • Demyelination (caution MS)
  • HF worsening
  • Drug-induced lupus
  • Allergic reactions (especially anti-chimeric infliximab)
  • Possible malignancy (lymphoma in young)

351.3.3.6 JAK Inhibitor Black Box

  • Cardiovascular events
  • Thrombotic events
  • Malignancy
  • Mortality
  • More in ≥ 50, smokers, RA history
  • Monitor: lipids, CBC, CK

351.3.3.7 S1P Modulator Side Effects

  • Bradyarrhythmia (first dose)
  • Macular edema
  • Lymphopenia
  • Liver enzymes
  • Infections

351.3.3.8 Strictureplasty (CD)

  • Preserve bowel
  • Alternative to resection for short strictures

351.3.3.9 Multidisciplinary Care

  • Gastroenterologist + colorectal surgeon + dietitian + IBD nurse + mental health + pharmacist

351.3.3.10 IBD + Cancer

  • ↑ CRC (long-standing colitis)
  • Lymphoma (especially with thiopurines)
  • Skin cancer (immunosuppression)
  • Surveillance

351.3.3.11 IBD Microbiome Therapies

  • FMT trials (mixed results)
  • Specific probiotics
  • Diet-based interventions (Crohn’s exclusive enteral nutrition pediatric)

351.3.3.12 Pediatric IBD

  • Higher proportion with early-onset
  • Growth failure concern
  • Specific pediatric trials
  • Aggressive early biologic often

351.3.4 Pearls

  • CD vs UC hallmark differences must memorize
  • PSC strongly UC-associated
  • Mesalamine + topical for distal UC
  • Top-down with early biologic for moderate-severe
  • Vedolizumab gut-selective (less systemic IS)
  • Anti-IL-23 selective (risankizumab, mirikizumab) newer
  • JAK inhibitors + S1P modulators for UC oral options
  • Pregnancy: continue most biologics; stop MTX
  • CRC surveillance 8-10 yr after onset
  • Vaccinate before biologic (esp live)