230.1 🎓 醫孞生版

230.1.0.1 📌 䞀頁重點

230.1.0.1.1 2 Subspecies
  • Trypanosoma brucei gambiense (W + C Africa) — slow, chronic, > 95% of human cases
  • Trypanosoma brucei rhodesiense (E + S Africa) — rapid, acute, sometimes fatal in weeks
230.1.0.1.2 Vector + Reservoir
  • Tsetse fly (Glossina spp.) — both subspecies
  • Reservoirs:
    • T. b. gambiense: humans primary (anthroponotic)
    • T. b. rhodesiense: cattle + wild animals (zoonotic)
230.1.0.1.3 Epidemiology (WHO 2024)
  • ~ 800-1000 reported cases/yr globally (mostly DRC)
  • WHO 2030 elimination of T. b. gambiense as public health problem (near)
  • 2024 trends: declining incidence
230.1.0.1.4 Clinical (2 Stages)
230.1.0.1.4.1 Stage 1: Hemolymphatic (Early)
  • Inoculation chancre at tsetse bite site (transient, often missed)
  • Fever (intermittent)
  • LAP (Winterbottom’s sign = posterior cervical LAP — pathognomonic for T. b. gambiense)
  • Hepatosplenomegaly
  • Anemia + thrombocytopenia
  • Itching, rash
  • Lasts months (gambiense) to weeks (rhodesiense)
230.1.0.1.4.2 Stage 2: Meningoencephalitic (Late / CNS)
  • Sleep disturbances (gives “sleeping sickness” name): hypersomnia daytime, insomnia night, sleep cycle reversal
  • Behavioral changes, apathy, depression, psychosis
  • Movement disorders (extrapyramidal + cerebellar)
  • Progressive neurological decline → coma → death without treatment
  • Months (gambiense) to weeks (rhodesiense)
230.1.0.1.5 Diagnosis
  • Card Agglutination Test for Trypanosomiasis (CATT) — screening for T. b. gambiense
  • Thick + thin blood smears, lymph node aspirate, CSF microscopy — direct visualization of trypomastigotes
  • CSF examination for staging:
    • Stage 2 if CSF WBC > 5 cells/µL or trypanosomes present
  • PCR + immunoassays — emerging
  • Card test for HAT (now widely available POC test)
230.1.0.1.6 Treatment (2024 Update)
230.1.0.1.6.1 T. b. gambiense (W + C Africa)
  • Stage 1: Fexinidazole (oral, 10 days) — replaces pentamidine in most settings
    • Alternative: pentamidine IM × 7d
  • Stage 2: Fexinidazole (oral, 10 days) — replaces NECT (nifurtimox-eflornithine combination therapy)
    • NECT (10-day eflornithine + 10-day nifurtimox) still in use some settings
  • Acoziborole (single-dose oral) — Phase 3 success 2024, regulatory submission ongoing; will revolutionize
230.1.0.1.6.2 T. b. rhodesiense (E + S Africa)
  • Stage 1: Suramin IV (no oral alternative yet)
  • Stage 2: Melarsoprol IV (arsenic-based, very toxic 5% encephalopathy mortality but reduces in disease)
  • Fexinidazole + acoziborole being trialed for rhodesiense
230.1.0.1.7 Prevention
  • Tsetse fly avoidance (long clothing, light colors, repellent)
  • Vector control (traps, insecticide-treated targets, drug-impregnated cattle)
  • Surveillance + active case finding + treatment

230.1.0.2 1⃣ Microbiology + Life Cycle

230.1.0.2.1 Trypanosoma brucei
  • Trypomastigote: extracellular flagellated form in blood/CSF
  • Epimastigote: in tsetse fly
  • Surface variant glycoprotein (VSG) — antigenic variation → continuous evasion → fever periods
230.1.0.2.2 Antigenic Variation
  • 1000 different VSG genes

  • Switch every few days
  • Wave of parasitemia → IgM response → switch → new wave
  • Drives chronic relapsing fever
230.1.0.2.3 Life Cycle
  1. Tsetse bite → trypomastigotes injected
  2. Multiply in blood + lymph (Stage 1)
  3. Cross blood-brain barrier → CNS (Stage 2)
  4. Tsetse takes blood meal → trypomastigotes ingested
  5. Transform to epimastigotes in tsetse → multiply → re-enter human

230.1.0.3 2⃣ Clinical Features

230.1.0.3.1 Inoculation Chancre
  • 5-15 days post-tsetse bite
  • Painful indurated nodule at bite site
  • Transient (1-3 weeks)
  • More common with T. b. rhodesiense
230.1.0.3.2 Stage 1: Hemolymphatic
230.1.0.3.2.1 T. b. gambiense (Chronic)
  • Months-years duration
  • Intermittent fever
  • Winterbottom’s sign: posterior cervical LAP — pathognomonic
  • Hepatosplenomegaly
  • Generalized LAP
  • Anemia + thrombocytopenia
  • Pruritus
  • Cardiac involvement uncommon
230.1.0.3.2.2 T. b. rhodesiense (Acute)
  • Weeks duration
  • High intermittent fever
  • LAP less prominent
  • Myocarditis prominent
  • Hepatosplenomegaly
  • Sometimes hemorrhagic complications
230.1.0.3.3 Stage 2: Meningoencephalitic
230.1.0.3.3.1 Sleep Disturbances
  • Reversal of sleep-wake cycle
  • Daytime hypersomnia, nighttime insomnia
  • Pathognomonic for HAT
230.1.0.3.3.2 Other CNS Features
  • Mental status changes: apathy, depression, psychosis
  • Movement disorders: tremor, ataxia, chorea, parkinsonism
  • Speech changes
  • Cranial nerve palsies
  • Seizures
  • Coma → death without treatment
230.1.0.3.4 Differential
  • Malaria (always rule out first)
  • HIV
  • Viral / bacterial meningitis
  • Encephalitis (other causes)
  • Other CNS protozoal infections

230.1.0.4 3⃣ Diagnosis

230.1.0.4.1 Screening (Asymptomatic in Endemic)
  • CATT (Card Agglutination Test for Trypanosomiasis) — T. b. gambiense
  • Reactive → confirmatory testing
230.1.0.4.2 Direct Microscopy
  • Thick + thin blood smears (Giemsa)
  • Trypomastigotes have undulating membrane + flagellum
  • Better sensitivity in T. b. rhodesiense (higher parasitemia)
  • T. b. gambiense often low parasitemia — multiple smears + concentration
230.1.0.4.3 Lymph Node Aspirate
  • Posterior cervical LN
  • High sensitivity for T. b. gambiense
  • Microscopy for trypomastigotes
230.1.0.4.4 Cerebrospinal Fluid (CSF)
  • Lumbar puncture for staging (essential for treatment selection)
  • Stage 2 if: WBC > 5 cells/µL or trypomastigotes present
  • Increased protein
  • IgM elevated
  • Direct microscopy for trypomastigotes
230.1.0.4.5 PCR
  • Sensitive
  • Species + subspecies identification
  • Reference labs
230.1.0.4.6 Card Test for HAT (Combo)
  • POC test (2017+)
  • Antibody detection
  • Used in active surveillance
230.1.0.4.7 Other Tests
  • ELISA, immunofluorescence
  • Loop-mediated isothermal amplification (LAMP)

230.1.0.5 4⃣ Treatment

230.1.0.5.1 T. b. gambiense Treatment Algorithm (2024)
230.1.0.5.1.1 Stage 1 (Hemolymphatic, CSF normal)
  • Fexinidazole PO 10 days (preferred 2019 WHO + 2024)
    • Day 1-4: 1800 mg PO bid
    • Day 5-10: 1200 mg PO bid
    • Take with food (better absorption)
  • Alternative: Pentamidine 4 mg/kg IM/IV daily × 7d (older, side effects)
230.1.0.5.1.2 Stage 2 (CNS Involvement)
  • Fexinidazole PO 10 days — increasingly first-line
  • Alternative: NECT (Nifurtimox-Eflornithine Combination Therapy)
    • Eflornithine 400 mg/kg/d IV × 7 days
    • Nifurtimox 15 mg/kg/d PO × 10 days
    • WHO previous standard
    • Effective but requires IV access + monitoring
230.1.0.5.1.3 Acoziborole (2024 Breakthrough)
  • Single-dose oral ~ 480 mg
  • Phase 3 trial 2024: efficacy + safety profile excellent
  • Regulatory submission EMA + WHO 2024+
  • Will revolutionize HAT treatment
230.1.0.5.2 T. b. rhodesiense Treatment
230.1.0.5.2.1 Stage 1
  • Suramin IV (no oral alternative yet)
  • 1 g IV at days 1, 3, 5, 14, 21
  • Side effects: nephrotoxicity, infusion reactions
230.1.0.5.2.2 Stage 2
  • Melarsoprol IV (arsenic-based)
  • 2.2 mg/kg IV daily × 10 days
  • Severe toxicity: encephalopathy (5% mortality), peripheral neuropathy, dermatitis
  • “Reactive encephalopathy” 2-5% in 1st week
  • High historical use but progressively replaced
  • Fexinidazole + acoziborole being trialed for rhodesiense (efficacy promising)
230.1.0.5.3 Treatment Considerations
  • Lumbar puncture before treatment for staging
  • Post-treatment LP at 6 months to confirm cure (CSF normalization)
  • Pregnancy: fexinidazole safe in 2nd-3rd trimester (1st trimester avoid)
  • Pediatric: weight-based fexinidazole
230.1.0.5.4 Supportive Care
  • Hospitalization for severe + Stage 2
  • Anticonvulsants for seizures
  • Glucose monitoring
  • Fluid + electrolyte management

230.1.0.6 5⃣ Prevention + Public Health

230.1.0.6.1 Personal Protection
  • Light-colored clothing (tsetse attracted to dark + blue)
  • Long sleeves + pants
  • DEET repellent
  • Avoiding tsetse habitats (riverside vegetation, savanna)
230.1.0.6.2 Vector Control
  • Tsetse traps + insecticide-treated targets
  • Sequential aerial spraying historical
  • Sterile insect technique (SIT) — Zanzibar success story
  • Drug-impregnated cattle (zoonotic rhodesiense control)
230.1.0.6.3 Surveillance + Case Detection
  • Active surveillance — mobile teams in endemic villages
  • CATT screening + microscopy
  • Treat detected cases → reduces reservoir
230.1.0.6.4 WHO 2030 Elimination Targets
  • T. b. gambiense: elimination as public health problem (< 1 case per 10,000 in endemic foci) — near
  • T. b. rhodesiense: zoonotic control
  • 2020s: dramatic case reduction (~ 800-1000/yr from 30,000+ early 2000s)
230.1.0.6.5 No Vaccine
  • Antigenic variation (VSG) makes vaccine difficult
  • Research ongoing but no candidates near clinical use